Drug Gene Type Source tamoxifen EBPL Ki=0.0028(uM) D1 PubChem tamoxifen EBP Ki=0.005(uM) D1 PubChem tamoxifen ESR2 Ki=0.0119(uM) D1 PubChem tamoxifen ESR1 Ki=0.0119(uM) D1 PubChem tamoxifen DHCR7 IC50=0.012(uM) D1 PubChem tamoxifen EBP IC50=0.012(uM) D1 PubChem tamoxifen SIGMAR1 IC50=0.021(uM) D1 PubChem tamoxifen ESR1 Ki=0.03119(uM) D1 PubChem tamoxifen ESR1 Ki=0.0344(uM) D1 PubChem tamoxifen ESR2 Ki=0.0344(uM) D1 PubChem tamoxifen ESR1 IC50=0.039(uM) D1 PubChem tamoxifen ESR1 IC50=0.042(uM) D1 PubChem tamoxifen ESR1 IC50=0.07(uM) D1 PubChem tamoxifen ESR1 IC50=0.1(uM) D1 PubChem tamoxifen ESR1 Ki=0.157(uM) D1 PubChem tamoxifen ESR2 Ki=0.157(uM) D1 PubChem tamoxifen ESR2 IC50=0.17(uM) D1 PubChem tamoxifen ESRRA IC50=0.2(uM) D1 PubChem tamoxifen HTR2C IC50=0.46(uM) D1 PubChem tamoxifen ESR1 IC50=0.5(uM) D1 PubChem tamoxifen ESR2 IC50=0.5(uM) D1 PubChem tamoxifen ESR2 IC50=0.58(uM) D1 PubChem tamoxifen ESR1 IC50=0.58(uM) D1 PubChem tamoxifen ESR1 IC50=0.622(uM) D1 PubChem tamoxifen ESR1 Potency=0.8765(uM) D1 PubChem tamoxifen ESR1 IC50=0.904(uM) D1 PubChem tamoxifen ESR2 IC50=0.904(uM) D1 PubChem tamoxifen TBXAS1 IC50=0.916(uM) D1 PubChem tamoxifen KCNH2 IC50=0.967(uM) D1 PubChem tamoxifen HTR6 Ki=1.041(uM) D1 PubChem tamoxifen DRD3 IC50=1.072(uM) D1 PubChem tamoxifen ESR1 Ratio Potency (uM)=1.14663(uM) D1 PubChem tamoxifen FYN IC50=1.195(uM) D1 PubChem tamoxifen GMNN Potency=1.2995(uM) D1 PubChem tamoxifen SLC6A2 IC50=1.472(uM) D1 PubChem tamoxifen ESR1 Potency=1.5484(uM) D1 PubChem tamoxifen KCNH2 IC50=1.58489(uM) D1 PubChem tamoxifen ESR2 EC50=1.66(uM) D1 PubChem tamoxifen SLC6A3 IC50=1.841(uM) D1 PubChem tamoxifen ESR1 Ratio Potency (uM)=1.87599(uM) D1 PubChem tamoxifen ADRA2A IC50=1.935(uM) D1 PubChem tamoxifen ESR1 IC50=2.0(uM) D1 PubChem tamoxifen ESR2 IC50=2.0(uM) D1 PubChem tamoxifen HTR2B IC50=2.084(uM) D1 PubChem tamoxifen SLC6A4 IC50=2.334(uM) D1 PubChem tamoxifen ESR1 EC50=2.54(uM) D1 PubChem tamoxifen CHRM5 IC50=2.585(uM) D1 PubChem tamoxifen HTR6 IC50=2.679(uM) D1 PubChem tamoxifen CHRM1 IC50=2.829(uM) D1 PubChem tamoxifen ERBB2 IC50=2.949(uM) D1 PubChem tamoxifen CHRM3 IC50=2.974(uM) D1 PubChem tamoxifen ADRA2B IC50=3.518(uM) D1 PubChem tamoxifen EGFR IC50=3.553(uM) D1 PubChem tamoxifen TACR2 IC50=3.67(uM) D1 PubChem tamoxifen ADORA3 IC50=3.701(uM) D1 PubChem tamoxifen CYP19A1 Potency=4.3541(uM) D1 PubChem tamoxifen PTGS1 IC50=4.391(uM) D1 PubChem tamoxifen HTR2A IC50=4.801(uM) D1 PubChem tamoxifen CHRM4 IC50=4.817(uM) D1 PubChem tamoxifen ADRA1D IC50=4.982(uM) D1 PubChem tamoxifen ADORA2A IC50=7.099(uM) D1 PubChem tamoxifen CYP19A1 Potency=7.6959(uM) D1 PubChem tamoxifen ADRB3 IC50=7.703(uM) D1 PubChem tamoxifen CHRM2 IC50=7.793(uM) D1 PubChem tamoxifen LCK IC50=8.033(uM) D1 PubChem tamoxifen DRD1 IC50=8.502(uM) D1 PubChem tamoxifen ESR1 Potency=8.6876(uM) D1 PubChem tamoxifen HRH2 IC50=9.396(uM) D1 PubChem tamoxifen ESR1 ER Potency (uM)=9.74769(uM) D1 PubChem tamoxifen DRD4 IC50=11.161(uM) D1 PubChem tamoxifen ESR1 IC50=11.3(uM) D1 PubChem tamoxifen ESR2 IC50=11.3(uM) D1 PubChem tamoxifen ESR1 ER Potency (uM)=13.1702(uM) D1 PubChem tamoxifen OPRD1 IC50=13.339(uM) D1 PubChem tamoxifen ESR1 Potency=13.6854(uM) D1 PubChem tamoxifen DRD2 IC50=13.885(uM) D1 PubChem tamoxifen OPRK1 IC50=15.629(uM) D1 PubChem tamoxifen TACR1 IC50=15.656(uM) D1 PubChem tamoxifen IDH1 Potency=16.3601(uM) D1 PubChem tamoxifen ADRB1 IC50=17.289(uM) D1 PubChem tamoxifen OPRM1 IC50=17.594(uM) D1 PubChem tamoxifen MC3R IC50=19.856(uM) D1 PubChem tamoxifen BDKRB2 IC50=20.356(uM) D1 PubChem tamoxifen ATXN2 Potency=22.3872(uM) D1 PubChem tamoxifen ADORA1 IC50=23.767(uM) D1 PubChem tamoxifen MC5R IC50=26.529(uM) D1 PubChem tamoxifen MC4R IC50=30.481(uM) D1 PubChem tamoxifen PPP3CA IC50=30.573(uM) D1 PubChem tamoxifen TP53 Potency=31.6228(uM) D1 PubChem tamoxifen UGT1A4 Km=32.0(uM) D1 PubChem tamoxifen BAZ2B Potency=35.4813(uM) D1 PubChem tamoxifen CBX1 Potency=35.4813(uM) D1 PubChem tamoxifen ATXN2 Potency=39.8107(uM) D1 PubChem tamoxifen PPARD Ratio Potency (uM)=54.941(uM) D1 PubChem tamoxifen ESR1 Potency=54.941(uM) D1 PubChem tamoxifen ESR1 Ratio Potency (uM)=54.9544(uM) D1 PubChem tamoxifen ESR1 Potency=77.4286(uM) D1 PubChem tamoxifen MLLT3 - D1 PubChem tamoxifen CYP19A1 - D1 PubChem tamoxifen CYP3A4 - D1 PubChem tamoxifen KCNQ1 - D1 PubChem tamoxifen PLD2 - D1 PubChem tamoxifen ESR2 - D1 PubChem tamoxifen STK33 - D1 PubChem tamoxifen CYP2C9 - D1 PubChem tamoxifen UBE2N - D1 PubChem tamoxifen ESR1 - D1 PubChem tamoxifen PLD1 - D1 PubChem tamoxifen CYP1A2 - D1 PubChem tamoxifen ESR1 Activity=None(Unspecified) D1 ChEMBL tamoxifen TP53 Potency=31622.8(nM) D1 ChEMBL tamoxifen ATXN2 Potency=22387.2(nM) D1 ChEMBL tamoxifen CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL tamoxifen CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL tamoxifen CYP1A2 Inhibition=None(Unspecified) D1 ChEMBL tamoxifen KDM4A Potency=44668.4(nM) D1 ChEMBL tamoxifen CBX1 Potency=35481.3(nM) D1 ChEMBL tamoxifen EHMT2 Potency=10000.0(nM) D1 ChEMBL tamoxifen ESR2 Activity=None(Unspecified) D1 ChEMBL tamoxifen PLD2 Activity=None(Unspecified) D1 ChEMBL tamoxifen BAZ2B Potency=35481.3(nM) D1 ChEMBL tamoxifen PLD1 Activity=None(Unspecified) D1 ChEMBL tamoxifen EHMT2 Potency=18887.6(nM) D1 ChEMBL tamoxifen ATXN2 Potency=39810.7(nM) D1 ChEMBL tamoxifen GMNN Potency=1299.5(nM) D1 ChEMBL tamoxifen EHMT2 Potency=12589.3(nM) D1 ChEMBL tamoxifen IDH1 Potency=16360.1(nM) D1 ChEMBL