Drug Gene Type Source 6-Thioguanine PAX8 AC50_uM=0.26(uM) D1 PubChem 6-Thioguanine PTGS1 IC50=0.601(uM) D1 PubChem 6-Thioguanine ESR1 Potency=0.7501(uM) D1 PubChem 6-Thioguanine TP53 Potency=1.0871(uM) D1 PubChem 6-Thioguanine HBB Potency=1.12202(uM) D1 PubChem 6-Thioguanine TDP1 Potency=1.1582(uM) D1 PubChem 6-Thioguanine PAX8 AC50_uM=1.18(uM) D1 PubChem 6-Thioguanine HPRT1 Km=1.7(uM) D1 PubChem 6-Thioguanine TDP1 Potency=1.8356(uM) D1 PubChem 6-Thioguanine TDP1 Potency=1.8837(uM) D1 PubChem 6-Thioguanine TDP1 Potency=2.1136(uM) D1 PubChem 6-Thioguanine IDH1 Potency=2.3109(uM) D1 PubChem 6-Thioguanine TDP1 Potency=2.5929(uM) D1 PubChem 6-Thioguanine TP53 Potency=2.6603(uM) D1 PubChem 6-Thioguanine TP53 Ratio Potency (uM)=2.66032(uM) D1 PubChem 6-Thioguanine TDP1 Potency=2.6609(uM) D1 PubChem 6-Thioguanine TP53 Potency=3.3491(uM) D1 PubChem 6-Thioguanine NFE2L2 Ratio Potency (uM)=3.71186(uM) D1 PubChem 6-Thioguanine NFE2L2 Potency=4.7326(uM) D1 PubChem 6-Thioguanine HBB Potency=5.0119(uM) D1 PubChem 6-Thioguanine NFE2L2 Ratio Potency (uM)=5.51527(uM) D1 PubChem 6-Thioguanine MAPK3 IC50=5.516(uM) D1 PubChem 6-Thioguanine HPRT1 Km=5.9(uM) D1 PubChem 6-Thioguanine NFE2L2 Ratio Potency (uM)=5.95797(uM) D1 PubChem 6-Thioguanine AR Potency=6.9167(uM) D1 PubChem 6-Thioguanine ESR1 ER Potency (uM)=8.41586(uM) D1 PubChem 6-Thioguanine AR Potency=10.6822(uM) D1 PubChem 6-Thioguanine AR Potency=16.9301(uM) D1 PubChem 6-Thioguanine ESR1 Ratio Potency (uM)=17.5753(uM) D1 PubChem 6-Thioguanine ESR1 Potency=18.9773(uM) D1 PubChem 6-Thioguanine ESR1 Potency=21.1317(uM) D1 PubChem 6-Thioguanine ADORA3 IC50=21.687(uM) D1 PubChem 6-Thioguanine NR3C1 Potency=23.9145(uM) D1 PubChem 6-Thioguanine AHR AhR Potency (uM)=28.1796(uM) D1 PubChem 6-Thioguanine NR3C1 Potency=30.111(uM) D1 PubChem 6-Thioguanine HBB Potency=31.6228(uM) D1 PubChem 6-Thioguanine HPGD Potency=35.4813(uM) D1 PubChem 6-Thioguanine NR3C1 Potency=43.6412(uM) D1 PubChem 6-Thioguanine AHR Potency=61.1306(uM) D1 PubChem 6-Thioguanine AHR AhR Potency (uM)=61.1306(uM) D1 PubChem 6-Thioguanine IMPDH1 - D1 PubChem 6-Thioguanine CYP19A1 - D1 PubChem 6-Thioguanine TNFRSF10B - D1 PubChem 6-Thioguanine TP53 Ratio Potency (uM)=None(uM) D1 PubChem 6-Thioguanine PAX8 - D1 PubChem 6-Thioguanine ITGA4 - D1 PubChem 6-Thioguanine IMPDH2 - D1 PubChem 6-Thioguanine MITF - D1 PubChem 6-Thioguanine HBB Potency=1122.02(nM) D1 ChEMBL 6-Thioguanine HBB Potency=31622.8(nM) D1 ChEMBL 6-Thioguanine PAX8 AC50=260.0(nM) D1 ChEMBL 6-Thioguanine KDM4A Potency=5623.4(nM) D1 ChEMBL 6-Thioguanine HPGD Potency=35481.3(nM) D1 ChEMBL 6-Thioguanine HBB Potency=5011.9(nM) D1 ChEMBL 6-Thioguanine EHMT2 Potency=2238.7(nM) D1 ChEMBL 6-Thioguanine IDH1 Potency=2310.9(nM) D1 ChEMBL 6-Thioguanine PAX8 AC50=1180.0(nM) D1 ChEMBL