Drug Gene Type Source doxepin KCNH2 IC50=6.45654(uM) D1 PubChem doxepin DRD1 Potency=2.2387(uM) D1 PubChem doxepin CYP2D6 Potency=3.1623(uM) D1 PubChem doxepin CYP2D6 Potency=3.9811(uM) D1 PubChem doxepin CYP2D6 Potency=15.8489(uM) D1 PubChem doxepin ALDH1A1 Potency=17.7828(uM) D1 PubChem doxepin CYP1A2 - D1 PubChem doxepin CYP2D6 - D1 PubChem doxepin ALDH1A1 Potency=17782.8(nM) D1 ChEMBL doxepin CYP2D6 AC50=15848.9(nM) D1 ChEMBL doxepin CYP2D6 AC50=3162.28(nM) D1 ChEMBL doxepin DRD1 Potency=2238.7(nM) D1 ChEMBL doxepin CYP2D6 Potency=3981.1(nM) D1 ChEMBL doxepin CYP2D6 Potency=15848.9(nM) D1 ChEMBL doxepin CYP2D6 Potency=3162.3(nM) D1 ChEMBL doxepin CYP1A2 AC50=15848.9(nM) D1 ChEMBL doxepin CYP2D6 AC50=3981.07(nM) D1 ChEMBL