Drug Gene Type Source cyclothiazide GRIA2 EC50=2.24(uM) D1 PubChem cyclothiazide GRIA4 EC50=3.8(uM) D1 PubChem cyclothiazide GRIA3 EC50=13.7(uM) D1 PubChem cyclothiazide GRIA1 EC50=19.8(uM) D1 PubChem cyclothiazide SLC12A3 - D1 PubChem cyclothiazide RECQL Potency=11220.2(nM) D1 ChEMBL