Drug Gene Type Source melphalan TDP1 Potency=0.2311(uM) D1 PubChem melphalan TDP1 Potency=0.2593(uM) D1 PubChem melphalan TDP1 Potency=0.5309(uM) D1 PubChem melphalan CYP3A4 Potency=3.1623(uM) D1 PubChem melphalan TP53 Potency=13.3332(uM) D1 PubChem melphalan ESR1 ER Potency (uM)=17.4947(uM) D1 PubChem melphalan TP53 Ratio Potency (uM)=18.8336(uM) D1 PubChem melphalan ESR1 Potency=23.3296(uM) D1 PubChem melphalan TP53 Potency=25.1189(uM) D1 PubChem melphalan TP53 Potency=26.1763(uM) D1 PubChem melphalan AR AR Potency (uM)=26.6032(uM) D1 PubChem melphalan RORC Potency=26.6032(uM) D1 PubChem melphalan AR Ratio Potency (uM)=26.8325(uM) D1 PubChem melphalan TP53 Ratio Potency (uM)=27.2003(uM) D1 PubChem melphalan AR Potency=29.8493(uM) D1 PubChem melphalan AR Potency=30.1065(uM) D1 PubChem melphalan ATAD5 ATAD5 Potency (uM)=31.0171(uM) D1 PubChem melphalan NR1H4 Potency=39.8107(uM) D1 PubChem melphalan TP53 Potency=39.8107(uM) D1 PubChem melphalan NFE2L2 Potency=42.1632(uM) D1 PubChem melphalan NR1I2 Potency=44.6684(uM) D1 PubChem melphalan NFE2L2 Potency=54.4827(uM) D1 PubChem melphalan STK33 - D1 PubChem melphalan MDM2 - D1 PubChem melphalan BARD1 - D1 PubChem melphalan ABCB1 - D1 PubChem melphalan MDM4 - D1 PubChem melphalan BRCA1 - D1 PubChem melphalan TP53 Potency=39810.7(nM) D1 ChEMBL melphalan NR1H4 Potency=39810.7(nM) D1 ChEMBL melphalan CYP3A4 Potency=3162.3(nM) D1 ChEMBL melphalan RORC Potency=26603.2(nM) D1 ChEMBL melphalan TP53 Potency=25118.9(nM) D1 ChEMBL melphalan NFE2L2 Potency=54482.7(nM) D1 ChEMBL melphalan EHMT2 Potency=7943.3(nM) D1 ChEMBL melphalan NFE2L2 Potency=42163.2(nM) D1 ChEMBL