Drug Gene Type Source tacrolimus MTOR IC50=0.00095(uM) D1 PubChem tacrolimus FKBP5 Ki=0.08(uM) D1 PubChem tacrolimus CYP3A4 IC50=1.0(uM) D1 PubChem tacrolimus TDP1 Potency=2.9855(uM) D1 PubChem tacrolimus TDP1 Potency=3.3498(uM) D1 PubChem tacrolimus AR Potency=16.9301(uM) D1 PubChem tacrolimus AR Ratio Potency (uM)=16.9301(uM) D1 PubChem tacrolimus FKBP1A - D1 PubChem