Drug Gene Type Source Fulvestrant ESR1 IC50=0.00021(uM) D1 PubChem Fulvestrant ESR2 IC50=0.00021(uM) D1 PubChem Fulvestrant ESR1 IC50=0.00047(uM) D1 PubChem Fulvestrant ESR1 Ki=0.000668(uM) D1 PubChem Fulvestrant ESR2 Ki=0.000668(uM) D1 PubChem Fulvestrant ESR2 Ki=0.000755(uM) D1 PubChem Fulvestrant ESR1 Ki=0.000755(uM) D1 PubChem Fulvestrant ESR1 Ki=0.00104(uM) D1 PubChem Fulvestrant ESR2 Ki=0.00139(uM) D1 PubChem Fulvestrant ESRRA IC50=0.002(uM) D1 PubChem Fulvestrant ESR1 IC50=0.004(uM) D1 PubChem Fulvestrant ESR2 IC50=0.004(uM) D1 PubChem Fulvestrant ESR1 IC50=0.0049(uM) D1 PubChem Fulvestrant ESR1 IC50=0.005(uM) D1 PubChem Fulvestrant ESR2 IC50=0.005(uM) D1 PubChem Fulvestrant ESR1 IC50=0.006(uM) D1 PubChem Fulvestrant EPHX2 IC50=0.006(uM) D1 PubChem Fulvestrant ESR1 ER Potency (uM)=0.00685199(uM) D1 PubChem Fulvestrant ESR2 IC50=0.007(uM) D1 PubChem Fulvestrant ESR2 Ki=0.00763(uM) D1 PubChem Fulvestrant ESR1 Ki=0.00763(uM) D1 PubChem Fulvestrant ESR2 IC50=0.0084(uM) D1 PubChem Fulvestrant ESR1 Potency=0.0086(uM) D1 PubChem Fulvestrant CYP19A1 Potency=0.0153(uM) D1 PubChem Fulvestrant ESR1 ER Potency (uM)=0.0219584(uM) D1 PubChem Fulvestrant ESR1 Ratio Potency (uM)=0.0254889(uM) D1 PubChem Fulvestrant EPHX2 Ki=0.026(uM) D1 PubChem Fulvestrant ESR1 Potency=0.0298(uM) D1 PubChem Fulvestrant ESR2 IC50=0.0441(uM) D1 PubChem Fulvestrant CYP19A1 Potency=0.0596(uM) D1 PubChem Fulvestrant ESR1 Ratio Potency (uM)=0.111001(uM) D1 PubChem Fulvestrant ESR1 Potency=0.6007(uM) D1 PubChem Fulvestrant NR1H4 IC50=0.79(uM) D1 PubChem Fulvestrant NR3C1 Potency=1.2294(uM) D1 PubChem Fulvestrant NR1I2 EC50=1.95(uM) D1 PubChem Fulvestrant ESR1 Potency=3.4648(uM) D1 PubChem Fulvestrant AR Ratio Potency (uM)=7.18374(uM) D1 PubChem Fulvestrant NFE2L2 Ratio Potency (uM)=17.2114(uM) D1 PubChem Fulvestrant ESR2 - D1 PubChem Fulvestrant EPHX2 - D1 PubChem Fulvestrant CYP19A1 - D1 PubChem Fulvestrant ESR1 - D1 PubChem Fulvestrant ESRRA - D1 PubChem Fulvestrant NR3C1 - D1 PubChem Fulvestrant NR1H4 - D1 PubChem Fulvestrant EPHX2 Inhibition=None(Unspecified) D1 ChEMBL Fulvestrant ESR1 Activity=None(Unspecified) D1 ChEMBL Fulvestrant ESR2 Activity=None(Unspecified) D1 ChEMBL Fulvestrant ESRRA Activity=None(Unspecified) D1 ChEMBL