Drug Gene Type Source Bexarotene RXRA EC50=0.0027(uM) D1 PubChem Bexarotene RXRA Kd=0.014(uM) D1 PubChem Bexarotene RXRA Ki=0.021(uM) D1 PubChem Bexarotene RXRA Kd=0.026(uM) D1 PubChem Bexarotene RXRA EC50=0.028(uM) D1 PubChem Bexarotene RXRA Ki=0.036(uM) D1 PubChem Bexarotene RXRA Kd=0.036(uM) D1 PubChem Bexarotene RXRA EC50=0.052(uM) D1 PubChem Bexarotene RXRG Ki=0.075(uM) D1 PubChem Bexarotene RXRA EC50=0.149(uM) D1 PubChem Bexarotene ESR1 Potency=3.7578(uM) D1 PubChem Bexarotene KAT2A Potency=6.3096(uM) D1 PubChem Bexarotene NR3C1 Potency=9.77(uM) D1 PubChem Bexarotene ESR1 Ratio Potency (uM)=10.9622(uM) D1 PubChem Bexarotene ESR1 Potency=17.3739(uM) D1 PubChem Bexarotene ESR1 ER Potency (uM)=18.8336(uM) D1 PubChem Bexarotene HSPB1 Ratio Potency (uM)=21.13(uM) D1 PubChem Bexarotene TP53 Potency=21.6899(uM) D1 PubChem Bexarotene USP1 Potency=22.3872(uM) D1 PubChem Bexarotene CYP19A1 Potency=61.1306(uM) D1 PubChem Bexarotene BLM Potency=68.0496(uM) D1 PubChem Bexarotene RXRB - D1 PubChem Bexarotene RXRG - D1 PubChem Bexarotene RXRA - D1 PubChem Bexarotene PPARG Ratio Potency (uM)=None(uM) D1 PubChem Bexarotene USP1 Potency=22387.2(nM) D1 ChEMBL Bexarotene KAT2A Potency=6309.6(nM) D1 ChEMBL Bexarotene RXRA Activity=None(Unspecified) D1 ChEMBL Bexarotene NR1H3 Activity=None(Unspecified) D1 ChEMBL Bexarotene BLM Potency=68049.6(nM) D1 ChEMBL