Drug Gene Type Source chlorpromazine DRD2 Ki=0.0012(uM) D1 PubChem chlorpromazine DRD3 Ki=0.003(uM) D1 PubChem chlorpromazine DRD3 Ki=0.00331(uM) D1 PubChem chlorpromazine HTR2A IC50=0.0034(uM) D1 PubChem chlorpromazine DRD3 Ki=0.0038(uM) D1 PubChem chlorpromazine HTR2A IC50=0.00385(uM) D1 PubChem chlorpromazine ADRA1D IC50=0.00399(uM) D1 PubChem chlorpromazine DRD2 Ki=0.00406(uM) D1 PubChem chlorpromazine HRH1 Ki=0.00425(uM) D1 PubChem chlorpromazine HTR2C IC50=0.00524(uM) D1 PubChem chlorpromazine HTR2A Ki=0.00589(uM) D1 PubChem chlorpromazine DRD3 Ki=0.0069(uM) D1 PubChem chlorpromazine HTR7 Ki=0.011(uM) D1 PubChem chlorpromazine HRH1 IC50=0.012(uM) D1 PubChem chlorpromazine DRD3 IC50=0.012(uM) D1 PubChem chlorpromazine DRD2 IC50=0.012(uM) D1 PubChem chlorpromazine HRH1 IC50=0.017(uM) D1 PubChem chlorpromazine SLC6A2 IC50=0.019(uM) D1 PubChem chlorpromazine CHRM5 IC50=0.025(uM) D1 PubChem chlorpromazine ADRA2B IC50=0.026(uM) D1 PubChem chlorpromazine HTR2C Ki=0.0302(uM) D1 PubChem chlorpromazine DRD4 Ki=0.03162(uM) D1 PubChem chlorpromazine SLC6A4 IC50=0.039(uM) D1 PubChem chlorpromazine HTR6 Ki=0.05(uM) D1 PubChem chlorpromazine HTR2B Ki=0.052(uM) D1 PubChem chlorpromazine DRD2 IC50=0.054(uM) D1 PubChem chlorpromazine HTR6 IC50=0.057(uM) D1 PubChem chlorpromazine HTR6 Ki=0.06026(uM) D1 PubChem chlorpromazine CHRM1 IC50=0.083(uM) D1 PubChem chlorpromazine DRD1 Ki=0.096(uM) D1 PubChem chlorpromazine SLC6A4 IC50=0.12(uM) D1 PubChem chlorpromazine HTR7 Ki=0.12023(uM) D1 PubChem chlorpromazine HTR2B IC50=0.126(uM) D1 PubChem chlorpromazine CHRM4 IC50=0.149(uM) D1 PubChem chlorpromazine CYP2D6 Potency=0.1585(uM) D1 PubChem chlorpromazine DRD5 Ki=0.172(uM) D1 PubChem chlorpromazine CHRM3 IC50=0.206(uM) D1 PubChem chlorpromazine DRD1 IC50=0.225(uM) D1 PubChem chlorpromazine ADRA2A IC50=0.352(uM) D1 PubChem chlorpromazine ADRA2C IC50=0.374(uM) D1 PubChem chlorpromazine CYP2D6 Potency=0.3981(uM) D1 PubChem chlorpromazine SIGMAR1 IC50=0.451(uM) D1 PubChem chlorpromazine AOX1 IC50=0.57(uM) D1 PubChem chlorpromazine CHRM2 IC50=0.652(uM) D1 PubChem chlorpromazine CALM1 Kd=1.24(uM) D1 PubChem chlorpromazine DRD4 IC50=1.365(uM) D1 PubChem chlorpromazine KCNH2 IC50=1.47(uM) D1 PubChem chlorpromazine KCNH2 IC50=1.47911(uM) D1 PubChem chlorpromazine HRH2 IC50=2.626(uM) D1 PubChem chlorpromazine SLC6A3 IC50=2.643(uM) D1 PubChem chlorpromazine KCNH2 IC50=5.8275(uM) D1 PubChem chlorpromazine CYP2D6 Ki=7.0(uM) D1 PubChem chlorpromazine MC5R IC50=7.617(uM) D1 PubChem chlorpromazine FYN IC50=8.68(uM) D1 PubChem chlorpromazine TDP1 Potency=10.0(uM) D1 PubChem chlorpromazine TP53 Potency=10.0(uM) D1 PubChem chlorpromazine OPRK1 IC50=11.082(uM) D1 PubChem chlorpromazine TDP1 Potency=11.2202(uM) D1 PubChem chlorpromazine THPO Potency=12.5893(uM) D1 PubChem chlorpromazine OPRM1 IC50=14.397(uM) D1 PubChem chlorpromazine MC4R IC50=15.204(uM) D1 PubChem chlorpromazine IDH1 Potency=15.8489(uM) D1 PubChem chlorpromazine ERBB2 IC50=19.366(uM) D1 PubChem chlorpromazine OPRD1 IC50=20.894(uM) D1 PubChem chlorpromazine TDP1 Potency=23.715(uM) D1 PubChem chlorpromazine MC3R IC50=24.343(uM) D1 PubChem chlorpromazine NR1H4 Potency=26.6011(uM) D1 PubChem chlorpromazine SLC22A1 IC50=27.0(uM) D1 PubChem chlorpromazine TACR2 IC50=27.195(uM) D1 PubChem chlorpromazine EGFR IC50=28.868(uM) D1 PubChem chlorpromazine HTR7 - D1 PubChem chlorpromazine CYP2C9 - D1 PubChem chlorpromazine HTR1A - D1 PubChem chlorpromazine CYP1A2 - D1 PubChem chlorpromazine CYP2D6 - D1 PubChem chlorpromazine MAPT - D1 PubChem chlorpromazine CYP3A4 - D1 PubChem chlorpromazine DRD2 - D1 PubChem chlorpromazine HTR6 - D1 PubChem chlorpromazine HTR2A - D1 PubChem chlorpromazine DRD4 - D1 PubChem chlorpromazine DRD3 - D1 PubChem chlorpromazine TP53 Ratio Potency (uM)=None(uM) D1 PubChem chlorpromazine HTR2C - D1 PubChem chlorpromazine CYP1A2 AC50=1000.0(nM) D1 ChEMBL chlorpromazine CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL chlorpromazine CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL chlorpromazine CYP2D6 AC50=158.49(nM) D1 ChEMBL chlorpromazine CYP2D6 Potency=398.1(nM) D1 ChEMBL chlorpromazine CYP2D6 Potency=158.5(nM) D1 ChEMBL chlorpromazine TP53 Potency=10000.0(nM) D1 ChEMBL chlorpromazine THPO Potency=12589.3(nM) D1 ChEMBL chlorpromazine CYP1A2 AC50=3981.07(nM) D1 ChEMBL chlorpromazine IDH1 Potency=15848.9(nM) D1 ChEMBL chlorpromazine CYP2D6 AC50=398.11(nM) D1 ChEMBL