Drug Gene Type Source diltiazem CYP3A4 Ki=0.1(uM) D1 PubChem diltiazem CYP3A4 IC50=1.8366(uM) D1 PubChem diltiazem CYP3A4 Potency=3.9811(uM) D1 PubChem diltiazem SLC22A1 IC50=12.4(uM) D1 PubChem diltiazem KCNH2 IC50=17.3(uM) D1 PubChem diltiazem KCNH2 IC50=17.378(uM) D1 PubChem diltiazem TDP1 Potency=26.6086(uM) D1 PubChem diltiazem ABCB1 IC50=42.658(uM) D1 PubChem diltiazem CYP1A2 - D1 PubChem diltiazem CYP3A4 - D1 PubChem diltiazem CYP2D6 - D1 PubChem diltiazem CYP2C19 - D1 PubChem diltiazem CYP2C9 - D1 PubChem diltiazem CYP2C19 Inhibition=None(Unspecified) D1 ChEMBL diltiazem CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL diltiazem CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL diltiazem CYP2D6 Inhibition=None(Unspecified) D1 ChEMBL diltiazem CYP1A2 Inhibition=None(Unspecified) D1 ChEMBL diltiazem CYP3A4 Potency=3981.1(nM) D1 ChEMBL diltiazem CYP3A4 AC50=3981.07(nM) D1 ChEMBL