Drug Gene Type Source pimozide KCNH2 IC50=0.00302(uM) D1 PubChem pimozide KCNH2 IC50=0.018(uM) D1 PubChem pimozide KCNH2 IC50=0.0182(uM) D1 PubChem pimozide KCNH2 Ki=0.042(uM) D1 PubChem pimozide KCNH2 IC50=0.05012(uM) D1 PubChem pimozide KCNH2 IC50=0.0546(uM) D1 PubChem pimozide KCNH2 IC50=0.05495(uM) D1 PubChem pimozide KCNH2 Potency=0.0562(uM) D1 PubChem pimozide OPRM1 IC50=0.372(uM) D1 PubChem pimozide HIF1A Potency=2.5119(uM) D1 PubChem pimozide CYP3A4 Potency=3.1623(uM) D1 PubChem pimozide CYP2D6 Potency=3.1623(uM) D1 PubChem pimozide OPRD1 IC50=3.76(uM) D1 PubChem pimozide CYP3A4 Potency=5.0119(uM) D1 PubChem pimozide HIF1A Potency=5.0119(uM) D1 PubChem pimozide NPSR1 Potency=6.3096(uM) D1 PubChem pimozide TDP1 Potency=6.6838(uM) D1 PubChem pimozide CYP2C19 Potency=10.0(uM) D1 PubChem pimozide XBP1 Absolute IC50 (XBP1)=10.0(uM) D1 PubChem pimozide CYP2D6 Potency=10.0(uM) D1 PubChem pimozide THPO Potency=10.0(uM) D1 PubChem pimozide ATAD5 Potency=11.5774(uM) D1 PubChem pimozide NPSR1 Potency=12.5893(uM) D1 PubChem pimozide AR Potency=13.8006(uM) D1 PubChem pimozide TDP1 Potency=14.581(uM) D1 PubChem pimozide TP53 Potency=15.8489(uM) D1 PubChem pimozide IDH1 Potency=16.3601(uM) D1 PubChem pimozide MTOR Potency=16.4816(uM) D1 PubChem pimozide RXRA Potency=17.7828(uM) D1 PubChem pimozide MPHOSPH8 Potency=22.3872(uM) D1 PubChem pimozide AR AR Potency (uM)=23.4203(uM) D1 PubChem pimozide TP53 Potency=25.1189(uM) D1 PubChem pimozide MAPK1 Potency=25.1189(uM) D1 PubChem pimozide TDP1 Potency=25.4789(uM) D1 PubChem pimozide CYP19A1 Potency=30.6379(uM) D1 PubChem pimozide ATXN2 Potency=31.6228(uM) D1 PubChem pimozide TDP1 Potency=32.076(uM) D1 PubChem pimozide PPARD Potency=33.4889(uM) D1 PubChem pimozide SLC22A2 IC50=34.2(uM) D1 PubChem pimozide PPARG Potency=34.6654(uM) D1 PubChem pimozide CBX1 Potency=35.4813(uM) D1 PubChem pimozide STK33 - D1 PubChem pimozide PIP4K2A Potency=None(uM) D1 PubChem pimozide MAP4K2 - D1 PubChem pimozide IL1B - D1 PubChem pimozide MMP14 EC50=None(uM) D1 PubChem pimozide DRD2 IC50=None(uM) D1 PubChem pimozide DRD2 - D1 PubChem pimozide DRD5 - D1 PubChem pimozide DRD1 - D1 PubChem pimozide HTR2A - D1 PubChem pimozide DRD4 - D1 PubChem pimozide DRD3 - D1 PubChem pimozide ADRB2 - D1 PubChem pimozide APAF1 - D1 PubChem pimozide NTSR1 - D1 PubChem pimozide CYP1A2 - D1 PubChem pimozide CYP2D6 - D1 PubChem pimozide MDM2 - D1 PubChem pimozide MDM4 - D1 PubChem pimozide CHRM1 - D1 PubChem pimozide ABCB1 - D1 PubChem pimozide HTR1A - D1 PubChem pimozide CACNA1H - D1 PubChem pimozide TP53 Potency=15848.9(nM) D1 ChEMBL pimozide KDM4A Potency=39810.7(nM) D1 ChEMBL pimozide CBX1 Potency=35481.3(nM) D1 ChEMBL pimozide MAPK1 Potency=25118.9(nM) D1 ChEMBL pimozide RXRA Potency=17782.8(nM) D1 ChEMBL pimozide CYP2D6 Potency=3162.3(nM) D1 ChEMBL pimozide CYP3A4 Potency=3162.3(nM) D1 ChEMBL pimozide THPO Potency=10000.0(nM) D1 ChEMBL pimozide NPSR1 Potency=6309.6(nM) D1 ChEMBL pimozide MPHOSPH8 Potency=22387.2(nM) D1 ChEMBL pimozide NPSR1 Potency=12589.3(nM) D1 ChEMBL pimozide CYP3A4 Potency=5011.9(nM) D1 ChEMBL pimozide CYP2D6 Potency=10000.0(nM) D1 ChEMBL pimozide CYP2C19 Potency=10000.0(nM) D1 ChEMBL pimozide XBP1 IC50=10000.0(nM) D1 ChEMBL pimozide ATAD5 Potency=11577.4(nM) D1 ChEMBL pimozide TP53 Potency=25118.9(nM) D1 ChEMBL pimozide MTOR Potency=16481.6(nM) D1 ChEMBL pimozide HIF1A Potency=5011.9(nM) D1 ChEMBL pimozide HIF1A Potency=2511.9(nM) D1 ChEMBL pimozide KCNH2 Potency=56.2(nM) D1 ChEMBL pimozide ATXN2 Potency=31622.8(nM) D1 ChEMBL pimozide CYP2D6 AC50=3162.28(nM) D1 ChEMBL pimozide IDH1 Potency=16360.1(nM) D1 ChEMBL