Drug Gene Type Source Amitriptyline hydrochloride ESR1 Ratio Potency (uM)=10.3502(uM) D1 PubChem Amitriptyline hydrochloride KCNH2 Potency=15.8489(uM) D1 PubChem Amitriptyline hydrochloride ALDH1A1 Potency=17.7828(uM) D1 PubChem Amitriptyline hydrochloride GNAS Potency=19.9526(uM) D1 PubChem Amitriptyline hydrochloride TDP1 Potency=23.715(uM) D1 PubChem Amitriptyline hydrochloride TDP1 Potency=26.6086(uM) D1 PubChem Amitriptyline hydrochloride ESR1 Potency=54.9477(uM) D1 PubChem Amitriptyline hydrochloride TP53 Potency=61.1306(uM) D1 PubChem Amitriptyline hydrochloride AR AR Potency (uM)=61.1306(uM) D1 PubChem Amitriptyline hydrochloride SLC6A2 - D1 PubChem Amitriptyline hydrochloride DRD1 - D1 PubChem Amitriptyline hydrochloride DRD2 - D1 PubChem Amitriptyline hydrochloride SLC6A4 - D1 PubChem Amitriptyline hydrochloride CHRM5 - D1 PubChem Amitriptyline hydrochloride CHRM4 - D1 PubChem Amitriptyline hydrochloride CHRM1 - D1 PubChem Amitriptyline hydrochloride TLR3 - D1 PubChem Amitriptyline hydrochloride ALDH1A1 Potency=17782.8(nM) D1 ChEMBL Amitriptyline hydrochloride KCNH2 Potency=15848.9(nM) D1 ChEMBL Amitriptyline hydrochloride GNAS Potency=19952.6(nM) D1 ChEMBL