Drug Gene Type Source protriptyline ADORA3 IC50=0.0011(uM) D1 PubChem protriptyline SLC6A2 Kd=0.0014(uM) D1 PubChem protriptyline SLC6A2 IC50=0.0017(uM) D1 PubChem protriptyline SLC6A2 IC50=0.0021(uM) D1 PubChem protriptyline SLC6A2 Ki=0.0023(uM) D1 PubChem protriptyline SLC6A2 IC50=0.0025(uM) D1 PubChem protriptyline SLC6A2 IC50=0.0071(uM) D1 PubChem protriptyline SLC6A2 IC50=0.0091(uM) D1 PubChem protriptyline SLC6A2 IC50=0.017(uM) D1 PubChem protriptyline CYP2D6 Potency=3.9811(uM) D1 PubChem protriptyline NFKB1 Potency=8.9125(uM) D1 PubChem protriptyline THPO Potency=10.0(uM) D1 PubChem protriptyline DRD1 Potency=11.2202(uM) D1 PubChem protriptyline CYP2D6 Potency=15.8489(uM) D1 PubChem protriptyline CYP2D6 - D1 PubChem protriptyline MAPT - D1 PubChem protriptyline CYP2D6 AC50=3981.07(nM) D1 ChEMBL protriptyline CYP2D6 Potency=3981.1(nM) D1 ChEMBL protriptyline CYP2D6 Potency=15848.9(nM) D1 ChEMBL protriptyline THPO Potency=10000.0(nM) D1 ChEMBL protriptyline DRD1 Potency=11220.2(nM) D1 ChEMBL protriptyline HSD17B10 Potency=12589.3(nM) D1 ChEMBL protriptyline NFKB1 Potency=8912.5(nM) D1 ChEMBL protriptyline CYP2D6 AC50=15848.9(nM) D1 ChEMBL