Drug Gene Type Source orphenadrine CHRM5 IC50=0.028(uM) D1 PubChem orphenadrine CHRM4 IC50=0.125(uM) D1 PubChem orphenadrine CHRM1 IC50=0.148(uM) D1 PubChem orphenadrine CHRM3 IC50=0.175(uM) D1 PubChem orphenadrine CHRM2 IC50=0.376(uM) D1 PubChem orphenadrine CYP2D6 IC50=0.4(uM) D1 PubChem orphenadrine HTR2A IC50=0.436(uM) D1 PubChem orphenadrine SLC6A4 IC50=0.458(uM) D1 PubChem orphenadrine HTR2C IC50=0.534(uM) D1 PubChem orphenadrine KCNH2 IC50=0.85114(uM) D1 PubChem orphenadrine HTR6 IC50=1.121(uM) D1 PubChem orphenadrine HRH1 IC50=1.241(uM) D1 PubChem orphenadrine ADRA2B IC50=1.895(uM) D1 PubChem orphenadrine ADRA2A IC50=2.156(uM) D1 PubChem orphenadrine SLC22A2 IC50=2.5(uM) D1 PubChem orphenadrine SLC6A2 IC50=2.666(uM) D1 PubChem orphenadrine HTR2B IC50=3.391(uM) D1 PubChem orphenadrine HRH2 IC50=6.961(uM) D1 PubChem orphenadrine SLC22A1 IC50=12.6(uM) D1 PubChem