Drug Gene Type Source loratadine CYP2C19 IC50=0.016(uM) D1 PubChem loratadine KCNH2 IC50=0.16982(uM) D1 PubChem loratadine HRH1 IC50=0.17(uM) D1 PubChem loratadine KCNH2 IC50=0.173(uM) D1 PubChem loratadine KCNH2 IC50=0.17378(uM) D1 PubChem loratadine HTR2B IC50=0.245(uM) D1 PubChem loratadine HRH1 IC50=0.29(uM) D1 PubChem loratadine CYP2C19 Potency=0.3981(uM) D1 PubChem loratadine HRH1 Ki=0.414(uM) D1 PubChem loratadine TDP1 Potency=2.6609(uM) D1 PubChem loratadine NR1I2 EC50=3.0(uM) D1 PubChem loratadine NR1H4 IC50=3.07(uM) D1 PubChem loratadine NFE2L2 Ratio Potency (uM)=6.18824(uM) D1 PubChem loratadine NFE2L2 Ratio Potency (uM)=6.60073(uM) D1 PubChem loratadine NPSR1 Potency=7.9433(uM) D1 PubChem loratadine TDP1 Potency=11.8856(uM) D1 PubChem loratadine NPSR1 Potency=12.5893(uM) D1 PubChem loratadine TDP1 Potency=12.9953(uM) D1 PubChem loratadine PPARG Potency=13.3322(uM) D1 PubChem loratadine TDP1 Potency=14.9631(uM) D1 PubChem loratadine HIF1A Potency=15.8489(uM) D1 PubChem loratadine CYP2C9 Potency=15.8489(uM) D1 PubChem loratadine AR Potency=17.3739(uM) D1 PubChem loratadine MAPK1 Potency=19.9526(uM) D1 PubChem loratadine TDP1 Potency=20.5962(uM) D1 PubChem loratadine ESR1 Ratio Potency (uM)=22.5767(uM) D1 PubChem loratadine GMNN Potency=23.1093(uM) D1 PubChem loratadine TP53 Ratio Potency (uM)=23.7101(uM) D1 PubChem loratadine TP53 Potency=23.7101(uM) D1 PubChem loratadine ESR1 Potency=26.8325(uM) D1 PubChem loratadine AR AR Potency (uM)=27.644(uM) D1 PubChem loratadine CYP2D6 Potency=31.6228(uM) D1 PubChem loratadine KCNH2 IC50=39.0866(uM) D1 PubChem loratadine TSHR Potency=39.8107(uM) D1 PubChem loratadine PPARD Ratio Potency (uM)=59.3239(uM) D1 PubChem loratadine AR Potency=61.1306(uM) D1 PubChem loratadine TP53 Potency=61.1306(uM) D1 PubChem loratadine ESR1 Potency=61.1306(uM) D1 PubChem loratadine ESR1 ER Potency (uM)=61.1306(uM) D1 PubChem loratadine TP53 Ratio Potency (uM)=66.0073(uM) D1 PubChem loratadine HRH1 - D1 PubChem loratadine PHOSPHO1 IC50=None(uM) D1 PubChem loratadine PPARG - D1 PubChem loratadine CACNA1H - D1 PubChem loratadine DRD3 - D1 PubChem loratadine CYP2C9 - D1 PubChem loratadine HIF1A Potency=15848.9(nM) D1 ChEMBL loratadine CYP2D6 Potency=31622.8(nM) D1 ChEMBL loratadine CYP2C9 Potency=15848.9(nM) D1 ChEMBL loratadine NPSR1 Potency=7943.3(nM) D1 ChEMBL loratadine NPSR1 Potency=12589.3(nM) D1 ChEMBL loratadine TSHR Potency=39810.7(nM) D1 ChEMBL loratadine MAPK1 Potency=19952.6(nM) D1 ChEMBL loratadine GMNN Potency=23109.3(nM) D1 ChEMBL loratadine CYP2C19 Potency=398.1(nM) D1 ChEMBL loratadine CYP2C9 AC50=15848.9(nM) D1 ChEMBL