Drug Gene Type Source loperamide OPRM1 Ki=0.00053(uM) D1 PubChem loperamide OPRM1 IC50=0.00145(uM) D1 PubChem loperamide CYP2D6 Potency=0.0158(uM) D1 PubChem loperamide SIGMAR1 IC50=0.628(uM) D1 PubChem loperamide OPRD1 IC50=0.896(uM) D1 PubChem loperamide TSHR Potency=1.2589(uM) D1 PubChem loperamide DRD3 IC50=1.337(uM) D1 PubChem loperamide CYP2D6 IC50=2.0(uM) D1 PubChem loperamide SLC6A4 IC50=2.202(uM) D1 PubChem loperamide ADRB2 IC50=3.005(uM) D1 PubChem loperamide HRH2 IC50=3.081(uM) D1 PubChem loperamide OPRK1 IC50=3.125(uM) D1 PubChem loperamide HTR2B IC50=4.105(uM) D1 PubChem loperamide CYP3A4 Potency=5.0119(uM) D1 PubChem loperamide TEK Kd=5.9(uM) D1 PubChem loperamide TDP1 Potency=6.6838(uM) D1 PubChem loperamide TDP1 Potency=8.4144(uM) D1 PubChem loperamide TDP1 Potency=9.7264(uM) D1 PubChem loperamide CYP2D6 Potency=10.0(uM) D1 PubChem loperamide MTOR Potency=13.0918(uM) D1 PubChem loperamide MTOR Potency=18.4927(uM) D1 PubChem loperamide SLC22A1 IC50=23.7(uM) D1 PubChem loperamide TDP1 Potency=23.715(uM) D1 PubChem loperamide CYP2D6 Potency=25.1189(uM) D1 PubChem loperamide CYP19A1 Potency=26.6032(uM) D1 PubChem loperamide AR Potency=26.6032(uM) D1 PubChem loperamide TP53 Potency=31.6228(uM) D1 PubChem loperamide CYP2D6 - D1 PubChem loperamide PDE4B - D1 PubChem loperamide TEK - D1 PubChem loperamide STK33 - D1 PubChem loperamide TEK Activity=None(Unspecified) D1 ChEMBL loperamide CYP2D6 Potency=25118.9(nM) D1 ChEMBL loperamide CYP3A4 Potency=5011.9(nM) D1 ChEMBL loperamide CYP2D6 AC50=25118.9(nM) D1 ChEMBL loperamide CYP2D6 Potency=15.8(nM) D1 ChEMBL loperamide TP53 Potency=31622.8(nM) D1 ChEMBL loperamide TSHR Potency=1258.9(nM) D1 ChEMBL loperamide CYP2D6 Potency=10000.0(nM) D1 ChEMBL loperamide MTOR Potency=13091.8(nM) D1 ChEMBL loperamide MTOR Potency=18492.7(nM) D1 ChEMBL loperamide CYP2D6 AC50=15.85(nM) D1 ChEMBL loperamide CYP2D6 AC50=10000.0(nM) D1 ChEMBL