Drug Gene Type Source labetalol ADRB1 IC50=0.01(uM) D1 PubChem labetalol ADRB2 IC50=0.016(uM) D1 PubChem labetalol ADRA1D IC50=0.521(uM) D1 PubChem labetalol CYP2D6 IC50=0.8(uM) D1 PubChem labetalol SLC6A3 IC50=1.607(uM) D1 PubChem labetalol SIGMAR1 IC50=1.815(uM) D1 PubChem labetalol HTR2B IC50=3.037(uM) D1 PubChem labetalol SLC6A2 IC50=3.354(uM) D1 PubChem labetalol CYP1A2 - D1 PubChem labetalol CYP2D6 - D1 PubChem labetalol CYP3A4 - D1 PubChem labetalol CYP2C19 - D1 PubChem labetalol CYP2C9 - D1 PubChem labetalol HPSE - D1 PubChem labetalol CYP2C19 Inhibition=None(Unspecified) D1 ChEMBL labetalol CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL labetalol CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL labetalol CYP1A2 Inhibition=None(Unspecified) D1 ChEMBL labetalol CYP2D6 Inhibition=None(Unspecified) D1 ChEMBL labetalol HPSE Activity=None(Unspecified) D1 ChEMBL