Drug Gene Type Source imipramine SLC6A4 Ki=0.00077(uM) D1 PubChem imipramine SLC6A4 IC50=0.0011(uM) D1 PubChem imipramine SLC6A4 IC50=0.002(uM) D1 PubChem imipramine SLC6A4 IC50=0.0035(uM) D1 PubChem imipramine ADORA3 IC50=0.0044(uM) D1 PubChem imipramine SLC6A4 IC50=0.0068(uM) D1 PubChem imipramine SLC6A4 IC50=0.0069(uM) D1 PubChem imipramine SLC6A4 IC50=0.0073(uM) D1 PubChem imipramine SLC6A4 IC50=0.008(uM) D1 PubChem imipramine HRH1 IC50=0.027(uM) D1 PubChem imipramine SLC6A4 IC50=0.029(uM) D1 PubChem imipramine SLC6A2 IC50=0.074(uM) D1 PubChem imipramine HTR2A IC50=0.22(uM) D1 PubChem imipramine DRD2 IC50=0.41(uM) D1 PubChem imipramine SLC22A2 IC50=0.6(uM) D1 PubChem imipramine KCNH2 IC50=3.38844(uM) D1 PubChem imipramine KCNH2 IC50=3.4(uM) D1 PubChem imipramine CYP2D6 Potency=6.3096(uM) D1 PubChem imipramine SLC47A1 IC50=10.0(uM) D1 PubChem imipramine DRD1 Potency=14.1254(uM) D1 PubChem imipramine SLC22A1 IC50=17.1(uM) D1 PubChem imipramine CYP2D6 Potency=25.1189(uM) D1 PubChem imipramine SLC6A3 IC50=25.6(uM) D1 PubChem imipramine TDP1 Potency=29.8554(uM) D1 PubChem imipramine SLC22A1 IC50=37.0(uM) D1 PubChem imipramine CYP2D6 - D1 PubChem imipramine CYP3A4 - D1 PubChem imipramine CYP2C19 - D1 PubChem imipramine CYP2C9 - D1 PubChem imipramine CYP1A2 - D1 PubChem imipramine CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL imipramine CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL imipramine CYP2C19 Inhibition=None(Unspecified) D1 ChEMBL imipramine CYP1A2 Inhibition=None(Unspecified) D1 ChEMBL imipramine CYP2D6 Inhibition=None(Unspecified) D1 ChEMBL imipramine CYP2D6 AC50=25118.9(nM) D1 ChEMBL imipramine DRD1 Potency=14125.4(nM) D1 ChEMBL imipramine CYP2D6 AC50=6309.57(nM) D1 ChEMBL imipramine CYP2D6 Potency=6309.6(nM) D1 ChEMBL imipramine CYP2D6 Potency=25118.9(nM) D1 ChEMBL imipramine EHMT2 Potency=25118.9(nM) D1 ChEMBL