Drug Gene Type Source hexachlorophene MAPK14 IC50=0.0876(uM) D1 PubChem hexachlorophene MAPK1 IC50=0.196(uM) D1 PubChem hexachlorophene ADORA3 IC50=0.6389(uM) D1 PubChem hexachlorophene PTGS2 IC50=0.6443(uM) D1 PubChem hexachlorophene EGFR IC50=0.7486(uM) D1 PubChem hexachlorophene HSP90AA1 AC50_uM=0.77(uM) D1 PubChem hexachlorophene ESR1 Potency=0.7743(uM) D1 PubChem hexachlorophene MCL1 Absolute IC50=0.86(uM) D1 PubChem hexachlorophene GMNN Potency=0.92(uM) D1 PubChem hexachlorophene RORC Potency=1.0591(uM) D1 PubChem hexachlorophene CYP2C19 IC50=1.2265(uM) D1 PubChem hexachlorophene CYP1A2 IC50=1.3133(uM) D1 PubChem hexachlorophene ADORA2A IC50=1.6138(uM) D1 PubChem hexachlorophene AR Potency=1.7376(uM) D1 PubChem hexachlorophene TSHR Potency=2.1331(uM) D1 PubChem hexachlorophene ESR1 IC50=2.16156(uM) D1 PubChem hexachlorophene AR Potency=2.1624(uM) D1 PubChem hexachlorophene LCK IC50=2.4325(uM) D1 PubChem hexachlorophene MAPK3 IC50=2.4844(uM) D1 PubChem hexachlorophene TDP1 Potency=2.5929(uM) D1 PubChem hexachlorophene PARK2 Potency=2.8184(uM) D1 PubChem hexachlorophene ACHE IC50=3.0149(uM) D1 PubChem hexachlorophene TBXAS1 IC50=3.087(uM) D1 PubChem hexachlorophene USP2 Potency=3.1623(uM) D1 PubChem hexachlorophene TDP1 Potency=3.2643(uM) D1 PubChem hexachlorophene PAX8 AC50_uM=3.3(uM) D1 PubChem hexachlorophene ERBB2 IC50=3.3188(uM) D1 PubChem hexachlorophene FYN IC50=3.478(uM) D1 PubChem hexachlorophene TACR2 IC50=4.1392(uM) D1 PubChem hexachlorophene TDP1 Potency=4.2172(uM) D1 PubChem hexachlorophene SLC6A4 IC50=4.3494(uM) D1 PubChem hexachlorophene HTR2C IC50=4.6042(uM) D1 PubChem hexachlorophene ESR1 Ratio Potency (uM)=4.61196(uM) D1 PubChem hexachlorophene TDP1 Potency=4.7318(uM) D1 PubChem hexachlorophene ALOX15 Potency=5.0119(uM) D1 PubChem hexachlorophene USP2 Potency=5.2119(uM) D1 PubChem hexachlorophene CYP19A1 Potency=5.4316(uM) D1 PubChem hexachlorophene AR Potency=5.4483(uM) D1 PubChem hexachlorophene VCP IC50=5.488(uM) D1 PubChem hexachlorophene ADRA2A IC50=5.4965(uM) D1 PubChem hexachlorophene HTT Potency=5.6234(uM) D1 PubChem hexachlorophene SMAD3 Potency=5.6234(uM) D1 PubChem hexachlorophene SUMO1 IC50_Mean=5.63(uM) D1 PubChem hexachlorophene FASN IC50=5.68(uM) D1 PubChem hexachlorophene HTR2B IC50=5.6947(uM) D1 PubChem hexachlorophene IDH1 Potency=5.8048(uM) D1 PubChem hexachlorophene CYP19A1 Potency=6.1131(uM) D1 PubChem hexachlorophene AR AR Potency (uM)=6.70808(uM) D1 PubChem hexachlorophene NFE2L2 Potency=6.859(uM) D1 PubChem hexachlorophene ADRA2C IC50=6.9754(uM) D1 PubChem hexachlorophene FASN IC50=7.79(uM) D1 PubChem hexachlorophene TP53 Potency=7.9433(uM) D1 PubChem hexachlorophene SUMO2 IC50_Mean=8.49(uM) D1 PubChem hexachlorophene TP53 Potency=9.659(uM) D1 PubChem hexachlorophene NPY1R EC50=9.796(uM) D1 PubChem hexachlorophene ALOX15B Potency=10.0(uM) D1 PubChem hexachlorophene TSHR Potency=10.0(uM) D1 PubChem hexachlorophene CYP19A1 Potency=10.5909(uM) D1 PubChem hexachlorophene AR Potency=10.6822(uM) D1 PubChem hexachlorophene TP53 Potency=12.5893(uM) D1 PubChem hexachlorophene KAT2A Potency=12.5893(uM) D1 PubChem hexachlorophene TP53 Potency=13.3332(uM) D1 PubChem hexachlorophene AR Potency=13.3332(uM) D1 PubChem hexachlorophene HSPB1 Ratio Potency (uM)=13.8022(uM) D1 PubChem hexachlorophene HSPB1 Ratio Potency (uM)=14.3957(uM) D1 PubChem hexachlorophene NFE2L2 Potency=14.581(uM) D1 PubChem hexachlorophene MCL1 IC50=14.8332(uM) D1 PubChem hexachlorophene SUMO2 IC50_Mean=15.8(uM) D1 PubChem hexachlorophene CYP3A4 Potency=15.8489(uM) D1 PubChem hexachlorophene GMNN Potency=16.3601(uM) D1 PubChem hexachlorophene EIF4G1 Absolute IC50=17.9374(uM) D1 PubChem hexachlorophene MAPT Potency=19.9526(uM) D1 PubChem hexachlorophene GALK1 Potency=21.1143(uM) D1 PubChem hexachlorophene TP53 Ratio Potency (uM)=21.1317(uM) D1 PubChem hexachlorophene PLK1 Potency=21.1923(uM) D1 PubChem hexachlorophene PPARD Potency=21.8216(uM) D1 PubChem hexachlorophene TDP1 Potency=23.1093(uM) D1 PubChem hexachlorophene HSPA8 IC50=27.4(uM) D1 PubChem hexachlorophene POLB Potency=28.1838(uM) D1 PubChem hexachlorophene TP53 Ratio Potency (uM)=30.5444(uM) D1 PubChem hexachlorophene RAPGEF4 Potency=31.6228(uM) D1 PubChem hexachlorophene USP1 Potency=31.6228(uM) D1 PubChem hexachlorophene HPGD Potency=35.4813(uM) D1 PubChem hexachlorophene POLH Potency=44.6684(uM) D1 PubChem hexachlorophene VDR Potency=44.6684(uM) D1 PubChem hexachlorophene THRB Potency=44.6684(uM) D1 PubChem hexachlorophene BAZ2B Potency=50.1187(uM) D1 PubChem hexachlorophene HSPB1 Ratio Potency (uM)=52.3463(uM) D1 PubChem hexachlorophene TP53 Potency=54.4827(uM) D1 PubChem hexachlorophene PPARG Ratio Potency (uM)=54.9477(uM) D1 PubChem hexachlorophene TP53 Ratio Potency (uM)=61.1306(uM) D1 PubChem hexachlorophene PPARD Ratio Potency (uM)=61.5015(uM) D1 PubChem hexachlorophene RAPGEF3 Potency=70.7946(uM) D1 PubChem hexachlorophene USP1 Potency=79.4328(uM) D1 PubChem hexachlorophene KLF5 - D1 PubChem hexachlorophene TSHR - D1 PubChem hexachlorophene ESR1 - D1 PubChem hexachlorophene MC4R - D1 PubChem hexachlorophene CACNA1H - D1 PubChem hexachlorophene PPP1CA - D1 PubChem hexachlorophene MDM4 - D1 PubChem hexachlorophene CFTR - D1 PubChem hexachlorophene MDM2 - D1 PubChem hexachlorophene BARD1 - D1 PubChem hexachlorophene VCP - D1 PubChem hexachlorophene MITF - D1 PubChem hexachlorophene SIRT5 - D1 PubChem hexachlorophene KCNQ1 - D1 PubChem hexachlorophene NFKB1 - D1 PubChem hexachlorophene PTGER2 - D1 PubChem hexachlorophene EIF4H IC50=None(uM) D1 PubChem hexachlorophene FASN - D1 PubChem hexachlorophene PABPC1 IC50=None(uM) D1 PubChem hexachlorophene ATG4B - D1 PubChem hexachlorophene SAE1 IC50=None(uM) D1 PubChem hexachlorophene STAT3 - D1 PubChem hexachlorophene NLRP1 - D1 PubChem hexachlorophene SLC12A5 - D1 PubChem hexachlorophene CASP6 - D1 PubChem hexachlorophene CASP1 - D1 PubChem hexachlorophene ESR2 - D1 PubChem hexachlorophene SLC5A7 - D1 PubChem hexachlorophene STK33 - D1 PubChem hexachlorophene UBA2 IC50=None(uM) D1 PubChem hexachlorophene MRGPRX1 - D1 PubChem hexachlorophene PLA2G7 - D1 PubChem hexachlorophene HCRTR1 - D1 PubChem hexachlorophene NLRP3 - D1 PubChem hexachlorophene NR2E3 - D1 PubChem hexachlorophene EIF4G1 - D1 PubChem hexachlorophene ADAM10 - D1 PubChem hexachlorophene DRD1 - D1 PubChem hexachlorophene PRNP - D1 PubChem hexachlorophene NPY2R - D1 PubChem hexachlorophene PLA2G1B - D1 PubChem hexachlorophene NOD1 EC50=None(uM) D1 PubChem hexachlorophene UBE2I IC50=None(uM) D1 PubChem hexachlorophene PAFAH2 - D1 PubChem hexachlorophene STAT1 - D1 PubChem hexachlorophene SLC6A3 - D1 PubChem hexachlorophene MCL1 - D1 PubChem hexachlorophene PPME1 - D1 PubChem hexachlorophene PAX8 - D1 PubChem hexachlorophene BRCA1 - D1 PubChem hexachlorophene SUMO1 - D1 PubChem hexachlorophene ADRB2 - D1 PubChem hexachlorophene HSP90AA1 AC50=770.0(nM) D1 ChEMBL hexachlorophene POLH Potency=44668.4(nM) D1 ChEMBL hexachlorophene VDR Potency=44668.4(nM) D1 ChEMBL hexachlorophene THRB Potency=44668.4(nM) D1 ChEMBL hexachlorophene MAPT Potency=19952.6(nM) D1 ChEMBL hexachlorophene USP2 Potency=5211.9(nM) D1 ChEMBL hexachlorophene TP53 Potency=12589.3(nM) D1 ChEMBL hexachlorophene VCP IC50=5488.0(nM) D1 ChEMBL hexachlorophene NFE2L2 Potency=14581.0(nM) D1 ChEMBL hexachlorophene HTT Potency=5623.4(nM) D1 ChEMBL hexachlorophene SMAD3 Potency=5623.4(nM) D1 ChEMBL hexachlorophene KDM4A Potency=79432.8(nM) D1 ChEMBL hexachlorophene ALOX15 Potency=5011.9(nM) D1 ChEMBL hexachlorophene GZMB Inhibition=None(Unspecified) D1 ChEMBL hexachlorophene POLB Potency=28183.8(nM) D1 ChEMBL hexachlorophene MCL1 IC50=14833.2(nM) D1 ChEMBL hexachlorophene BAZ2B Potency=50118.7(nM) D1 ChEMBL hexachlorophene USP2 Potency=3162.3(nM) D1 ChEMBL hexachlorophene KAT2A Potency=12589.3(nM) D1 ChEMBL hexachlorophene CYP3A4 Potency=15848.9(nM) D1 ChEMBL hexachlorophene TSHR Potency=10000.0(nM) D1 ChEMBL hexachlorophene HSPA8 IC50=27400.0(nM) D1 ChEMBL hexachlorophene NPY1R EC50=9796.0(nM) D1 ChEMBL hexachlorophene GALK1 Potency=21114.3(nM) D1 ChEMBL hexachlorophene TSHR Potency=2133.1(nM) D1 ChEMBL hexachlorophene RORC Potency=1059.1(nM) D1 ChEMBL hexachlorophene TP53 Potency=7943.3(nM) D1 ChEMBL hexachlorophene FASN IC50=7790.0(nM) D1 ChEMBL hexachlorophene SUMO1 IC50=5630.0(nM) D1 ChEMBL hexachlorophene FASN IC50=5680.0(nM) D1 ChEMBL hexachlorophene HSPA1B IC50=19500.0(nM) D1 ChEMBL hexachlorophene HSD17B10 Potency=7943.3(nM) D1 ChEMBL hexachlorophene HPGD Potency=35481.3(nM) D1 ChEMBL hexachlorophene ESR1 IC50=2161.56(nM) D1 ChEMBL hexachlorophene ALOX15B Potency=10000.0(nM) D1 ChEMBL hexachlorophene GMNN Potency=16360.1(nM) D1 ChEMBL hexachlorophene GMNN Potency=920.0(nM) D1 ChEMBL hexachlorophene IDH1 Potency=5804.8(nM) D1 ChEMBL hexachlorophene HSPA1B IC50=19200.0(nM) D1 ChEMBL hexachlorophene NFE2L2 Potency=6859.0(nM) D1 ChEMBL hexachlorophene USP1 Potency=79432.8(nM) D1 ChEMBL hexachlorophene USP1 Potency=31622.8(nM) D1 ChEMBL hexachlorophene PAX8 AC50=3300.0(nM) D1 ChEMBL