Drug Gene Type Source GUANFACINE NISCH Ki=0.01901(uM) D1 PubChem GUANFACINE CYP2D6 Potency=0.1259(uM) D1 PubChem GUANFACINE ADRA2A IC50=0.134(uM) D1 PubChem GUANFACINE ADRA2B IC50=0.249(uM) D1 PubChem GUANFACINE CYP2C19 Potency=0.2512(uM) D1 PubChem GUANFACINE HTR2C IC50=1.453(uM) D1 PubChem GUANFACINE HTR2B IC50=2.098(uM) D1 PubChem GUANFACINE HTR2A IC50=3.014(uM) D1 PubChem GUANFACINE ADRA2C IC50=6.447(uM) D1 PubChem GUANFACINE CYP3A4 Potency=12.5893(uM) D1 PubChem GUANFACINE CYP2D6 - D1 PubChem GUANFACINE CYP2C19 - D1 PubChem GUANFACINE CYP3A4 - D1 PubChem GUANFACINE CYP3A4 AC50=12589.2(nM) D1 ChEMBL GUANFACINE CYP3A4 Potency=12589.3(nM) D1 ChEMBL GUANFACINE CYP2C19 Potency=251.2(nM) D1 ChEMBL GUANFACINE CYP2D6 Potency=125.9(nM) D1 ChEMBL GUANFACINE EHMT2 Potency=12589.3(nM) D1 ChEMBL GUANFACINE CYP2D6 AC50=125.89(nM) D1 ChEMBL GUANFACINE CYP2C19 AC50=251.19(nM) D1 ChEMBL