Drug Gene Type Source Rifampicin SLCO1B1 IC50=1.2(uM) D1 PubChem Rifampicin SLCO1B3 IC50=1.5(uM) D1 PubChem Rifampicin NR1I2 EC50=2.3(uM) D1 PubChem Rifampicin NR1I2 EC50=5.6(uM) D1 PubChem Rifampicin CASP1 IC50=8.319(uM) D1 PubChem Rifampicin ALB Kd=12.0(uM) D1 PubChem Rifampicin CYP51A1 IC50=30.0(uM) D1 PubChem Rifampicin NR1I2 - D1 PubChem Rifampicin CYP2C9 - D1 PubChem Rifampicin CYP1A2 - D1 PubChem Rifampicin CYP2C19 - D1 PubChem Rifampicin ABCB1 - D1 PubChem Rifampicin CYP2D6 - D1 PubChem Rifampicin CYP3A4 - D1 PubChem Rifampicin CYP2C19 Inhibition=None(Unspecified) D1 ChEMBL Rifampicin CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL Rifampicin NR1I2 Activity=None(Unspecified) D1 ChEMBL Rifampicin CYP2D6 Inhibition=None(Unspecified) D1 ChEMBL Rifampicin CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL Rifampicin CYP1A2 Inhibition=None(Unspecified) D1 ChEMBL