Drug Gene Type Source diphenhydramine HRH1 Ki=0.01479(uM) D1 PubChem diphenhydramine CHRM5 IC50=0.162(uM) D1 PubChem diphenhydramine HRH1 IC50=0.171(uM) D1 PubChem diphenhydramine CHRM1 IC50=0.346(uM) D1 PubChem diphenhydramine CHRM4 IC50=0.372(uM) D1 PubChem diphenhydramine CHRM3 IC50=0.647(uM) D1 PubChem diphenhydramine HTR2C IC50=0.98(uM) D1 PubChem diphenhydramine CHRM2 IC50=1.05(uM) D1 PubChem diphenhydramine HTR2B IC50=1.118(uM) D1 PubChem diphenhydramine HTR2A IC50=1.295(uM) D1 PubChem diphenhydramine KCNH2 IC50=2.5704(uM) D1 PubChem diphenhydramine SLC6A2 IC50=3.542(uM) D1 PubChem diphenhydramine CYP2D6 Potency=3.9811(uM) D1 PubChem diphenhydramine CYP2D6 Potency=12.5893(uM) D1 PubChem diphenhydramine KCNH2 IC50=26.9154(uM) D1 PubChem diphenhydramine KCNH2 IC50=31.859(uM) D1 PubChem diphenhydramine HRH4 Ki=42.658(uM) D1 PubChem diphenhydramine CYP2C19 - D1 PubChem diphenhydramine CYP2D6 - D1 PubChem diphenhydramine CYP1A2 - D1 PubChem diphenhydramine DRD3 - D1 PubChem diphenhydramine CYP3A4 - D1 PubChem diphenhydramine CHRM5 - D1 PubChem diphenhydramine CYP2C9 - D1 PubChem diphenhydramine CYP2C19 Inhibition=None(Unspecified) D1 ChEMBL diphenhydramine CYP2C9 Inhibition=None(Unspecified) D1 ChEMBL diphenhydramine CYP3A4 Inhibition=None(Unspecified) D1 ChEMBL diphenhydramine CYP2D6 Inhibition=None(Unspecified) D1 ChEMBL diphenhydramine CYP1A2 Inhibition=None(Unspecified) D1 ChEMBL diphenhydramine CYP2D6 Potency=12589.3(nM) D1 ChEMBL diphenhydramine CYP2D6 Potency=3981.1(nM) D1 ChEMBL diphenhydramine CYP2D6 AC50=12589.2(nM) D1 ChEMBL diphenhydramine CYP2D6 AC50=3981.07(nM) D1 ChEMBL